SU5205

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SU5205  纯度: 98.44%

SU5205 是 VEGFR2 (FLK-1) 的抑制剂，IC50 值为 9.6 μM。

SU5205

SU5205 Chemical Structure

CAS No. : 3476-86-6

规格 价格 是否有货 数量
10 mM * 1 mL in DMSO ￥550 In-stock
50 mg ￥500 In-stock
100 mg ￥800 In-stock
200 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

SU5205 相关产品

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生物活性

SU5205 is an inhibitor of VEGFR2 (FLK-1), with an IC50 of 9.6 μM[1].

IC50 & Target[1]

Flk-1

9.6 μM (IC50)

体外研究
(In Vitro)

SU5205 inhibits ligand-induced endothelial mitogenesis for VEGF with an IC50 of 5.1 μM[1].

上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

239.24

Formula

C15H10FNO
CAS 号

3476-86-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
溶解性数据
In Vitro: 

DMSO : 250 mg/mL (1044.98 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 4.1799 mL 20.8995 mL 41.7990 mL
5 mM 0.8360 mL 4.1799 mL 8.3598 mL
10 mM 0.4180 mL 2.0900 mL 4.1799 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Torsten K, et, al. Synthesis and radiopharmacological investigation of 3-[4′-[(18)F]fluorobenzylidene]indolin-2-one as possible tyrosine kinase inhibitor. Bioorg Med Chem. 2009 Nov 15; 17(22): 7732-42.

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