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GSK-5959 纯度: 98.29%
GSK-5959 是有效的、选择性的、细胞渗透性的 BRPF1 溴端结构域的抑制剂,其 IC50 值为 80 nM。
GSK-5959 Chemical Structure
CAS No. : 901245-65-6
规格 | 价格 | 是否有货 | 数量 |
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Free Sample (0.1-0.5 mg) | Apply now | ||
10 mM * 1 mL in DMSO | ¥990 | In-stock | |
5 mg | ¥900 | In-stock | |
10 mg | ¥1500 | In-stock | |
50 mg | ¥4500 | In-stock | |
100 mg | 询价 | ||
200 mg | 询价 |
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GSK-5959 相关产品
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生物活性 |
GSK-5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with an IC50 of ~ 80 nM[1]. |
IC50 & Target |
IC50: 80 nM (BRPF1)[1]. |
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体外研究 (In Vitro) |
GSK-5959 (3a) also displays selectivity over the closely related family members, BRPF2 (100-fold) and BRPF3 (>1000-fold)[2]. 上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
394.47 |
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Formula |
C22H26N4O3 |
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CAS 号 |
901245-65-6 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:
DMSO : 13 mg/mL (32.96 mM; Need ultrasonic and warming) 配制储备液
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请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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