BRD4 Inhibitor-16

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上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

BRD4 Inhibitor-16 

BRD4 Inhibitor-16 (Compound 4) 是溴域 4 (BRD4) 的有效抑制剂。 溴结构域 4 (BRD4) 的过表达通过调节组蛋白翻译后修饰与多种人类癌症密切相关。 BRD4 Inhibitor-16 是探索性研究 BRD4 抑制的有用工具，例如更好地了解 BRD4 抑制剂释放相关信息。

BRD4 Inhibitor-16

BRD4 Inhibitor-16 Chemical Structure

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生物活性

BRD4 Inhibitor-16 (Compound 4) is a potent inhibitor of bromodomain 4 (BRD4). Overexpression of bromodomain 4 (BRD4) is closely correlated with a variety of human cancers by regulating the histone post-translational modifications. BRD4 Inhibitor-16 represents a useful tool for explorative studies of BRD4 inhibition, such as an improved understanding of BRD4 inhibitor release-related information[1].

分子量

805.90

Formula

C42H43N7O8S
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Zhang H, et al. Activatable fluorescence molecular imaging and anti-tumor effects investigation of GSH-sensitive BRD4 ligands [published online ahead of print, 2022 Jan 25]. Bioorg Chem. 2022;120:105636.

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