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Umbralisib R-enantiomer (Synonyms: TGR-1202 R-enantiomer; RP5264 R-enantiomer) 纯度: 99.52%
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) 是 PI3Kδ 抑制剂,是 TGR-1202 活性较低的对映体。
Umbralisib R-enantiomer Chemical Structure
CAS No. : 1532533-69-9
规格 | 价格 | 是否有货 | 数量 |
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2 mg | ¥3500 | In-stock | |
5 mg | ¥7000 | In-stock | |
10 mg | 询价 | ||
50 mg | 询价 |
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Umbralisib R-enantiomer 相关产品
•相关化合物库:
- Bioactive Compound Library Plus
生物活性 |
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is a PI3Kδ inhibitor, which is the less active enantiomer of TGR-1202. |
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IC50 & Target[1] |
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体外研究 (In Vitro) |
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) (Formula A) exhibits a 50% inhibitory concentration (IC50) with respect to the δ type PI3-kinase that is at least 20-fold lower than the inhibitor’s IC50 with respect to the rest of the other PI3K isoforms (i.e., a, β, and γ)[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
571.55 |
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Formula |
C31H24F3N5O3 |
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CAS 号 |
1532533-69-9 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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参考文献 |
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