上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白,专注于信号通路和疾病研究领域。
Umbralisib R-enantiomer (Synonyms: TGR-1202 R-enantiomer; RP5264 R-enantiomer) 纯度: 99.52%
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) 是 PI3Kδ 抑制剂,是 TGR-1202 活性较低的对映体。
Umbralisib R-enantiomer Chemical Structure
CAS No. : 1532533-69-9
规格 | 价格 | 是否有货 | 数量 |
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2 mg | ¥3500 | In-stock | |
5 mg | ¥7000 | In-stock | |
10 mg | 询价 | ||
50 mg | 询价 |
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Umbralisib R-enantiomer 相关产品
•相关化合物库:
- Bioactive Compound Library Plus
生物活性 |
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is a PI3Kδ inhibitor, which is the less active enantiomer of TGR-1202. |
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IC50 & Target[1] |
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体外研究 (In Vitro) |
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) (Formula A) exhibits a 50% inhibitory concentration (IC50) with respect to the δ type PI3-kinase that is at least 20-fold lower than the inhibitor’s IC50 with respect to the rest of the other PI3K isoforms (i.e., a, β, and γ)[1]. 上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
571.55 |
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Formula |
C31H24F3N5O3 |
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CAS 号 |
1532533-69-9 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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参考文献 |
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