N-desmethyl Enzalutamide-d6(Synonyms: N-desmethyl MDV 3100-d6)

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白,专注于信号通路和疾病研究领域。

N-desmethyl Enzalutamide-d6 (Synonyms: N-desmethyl MDV 3100-d6)

N-desmethyl Enzalutamide D6 (N-desmethyl MDV 3100 D6) 是 N-desmethyl Enzalutamide 氘代物。N-desmethyl Enzalutamide 是Enzalutamide 的活性代谢产物。N-desmethyl Enzalutamide 具有与 Enzalutamide 相似的一级和二级药效功效,并在与 Enzalutamide 大致相同的血浆浓度下循环。

N-desmethyl Enzalutamide-d6(Synonyms: N-desmethyl MDV 3100-d6)

N-desmethyl Enzalutamide-d6 Chemical Structure

规格 是否有货
5 mg 询价
10 mg 询价

* Please select Quantity before adding items.

生物活性

N-desmethyl Enzalutamide D6 (N-desmethyl MDV 3100 D6) is a deuterium labeled N-desmethyl Enzalutamide. N-desmethyl Enzalutamide is an active metabolite of Enzalutamide. N-desmethyl Enzalutamide is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar potency to Enzalutamide and circulates at approximately the same plasma concentrations as enzalutamide[1].

IC50 & Target

Androgen-receptor[1]

分子量

456.45

Formula

C20H8D6F4N4O2S

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

参考文献
  • [1]. Gibbons JA, et al. Pharmacokinetic Drug Interaction Studies with Enzalutamide. Clin Pharmacokinet. 2015 Oct;54(10):1057-69.

所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务