Leelamine

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白,专注于信号通路和疾病研究领域。

Leelamine 

Leelamine 是大麻素受体 CB1CB2 的弱激动剂。Leelamine 也可以抑制丙酮酸脱氢酶激酶 (PDK)。Leelamine 具有抗肿瘤活性。

Leelamine

Leelamine Chemical Structure

CAS No. : 1446-61-3

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500 mg ¥500 In-stock
1 g ¥700 In-stock
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Leelamine 相关产品

相关化合物库:

  • Bioactive Compound Library Plus
  • GPCR/G Protein Compound Library
  • Kinase Inhibitor Library
  • Metabolism/Protease Compound Library
  • Neuronal Signaling Compound Library
  • Anti-Cancer Compound Library
  • Glycolysis Compound Library
  • Anti-Cancer Metabolism Compound Library
  • Mitochondria-Targeted Compound Library
  • Glucose Metabolism Compound Library

生物活性

Leelamine is a weak agonist of cannabinoid receptors CB1 and CB2. Leelamine also inhibits pyruvate dehydrogenase kinases (PDKs). Leelamine exhibits anti-tumor activity[1].

IC50 & Target[1]

CB1

 

CB2

 

分子量

285.47

Formula

C20H31N

CAS 号

1446-61-3

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

参考文献
  • [1]. Merarchi M, et, al. A Brief Overview of the Antitumoral Actions of Leelamine. Biomedicines. 2019 Jul 19;7(3):53.

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