PKG inhibitor peptide

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PKG inhibitor peptide  纯度: 98.15%

PKG inhibitor peptide 是一种 ATP 竞争性的 PKG 抑制剂，Ki 值为 86 μM。

PKG inhibitor peptide

PKG inhibitor peptide Chemical Structure

CAS No. : 82801-73-8

规格 价格 是否有货 数量
1 mg ￥900 In-stock
5 mg ￥2800 In-stock
10 mg ￥4500 In-stock
50 mg   询价  
100 mg   询价  

* Please select Quantity before adding items.

PKG inhibitor peptide 相关产品

•相关化合物库:

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  • Peptide Library

生物活性

PKG inhibitor peptide is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a Ki of 86 μM[1].

IC50 & Target

Ki: 86 μM (PKG)[1]
体外研究
(In Vitro)

Summary of experiments showing that intracellular dialysis of postsynaptic cells with PKG inhibitor PKG inhibitor peptide (1 mM) failed to alter the induction of long-term depression (CCh-LTD)[2].

Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

943.11

Formula

C38H74N18O10
CAS 号

82801-73-8
Sequence Shortening

RKRARKE
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -80°C 2 years
-20°C 1 year
In solvent -80°C 6 months
-20°C 1 month
溶解性数据
In Vitro: 

H2O : 100 mg/mL (106.03 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 1.0603 mL 5.3016 mL 10.6032 mL
5 mM 0.2121 mL 1.0603 mL 2.1206 mL
10 mM 0.1060 mL 0.5302 mL 1.0603 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Bhatnagar D, et al. Synthetic peptide analogues differentially alter the binding affinities of cyclic nucleotide dependent protein kinases for nucleotide substrates. Biochemistry. 1988 Mar 22;27(6):1988-94.

    [2]. Chiung-Chun Huang, et al. Activation of muscarinic acetylcholine receptors induces a nitric oxide-dependent long-term depression in rat medial prefrontal cortex. Cereb Cortex. 2010 Apr;20(4):982-96.

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