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1-Ethynylpyrene (Synonyms: 1-乙炔基芘) 纯度: 96.20%
1-Ethynylpyrene 是细胞色素 P450 1A1, 1A2 和 2B1 的抑制剂,IC50 分别为 0.18,0.32 和 0.04 μM。
1-Ethynylpyrene Chemical Structure
CAS No. : 34993-56-1
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10 mg | ¥800 | In-stock | |
50 mg | ¥2000 | In-stock | |
100 mg | ¥3400 | In-stock | |
200 mg | 询价 | ||
500 mg | 询价 |
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1-Ethynylpyrene 相关产品
•相关化合物库:
- Covalent Screening Library Plus
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- Anti-Aging Compound Library
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- Oxygen Sensing Compound Library
生物活性 |
1-Ethynylpyrene is an aryl acetylenic inhibitor of cytochromes P450 1A1, 1A2, and 2B1 with IC50s of 0.18, 0.32, and 0.04 μM, respectively[1]. |
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体外研究 (In Vitro) |
1-Ethynylpyrene exhibits activity against P450 1A2, and 2B1 with Kis of 0.32 and 0.04 μM, respectively[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
226.27 |
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Formula |
C18H10 |
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CAS 号 |
34993-56-1 |
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中文名称 |
1-乙炔基芘 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:
DMSO : 9.09 mg/mL (40.17 mM; ultrasonic and warming and heat to 60°C) 配制储备液
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请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用; 以下溶剂前显示的百
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参考文献 |
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