上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白,专注于信号通路和疾病研究领域。
PSI-697 (Synonyms: P-Selectin Inhibitor) 纯度: 99.70%
PSI-697 是一种口服的 P-selectin 抑制剂,IC50 值为 125 μM。
PSI-697 Chemical Structure
CAS No. : 851546-61-7
规格 | 价格 | 是否有货 | 数量 |
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10 mM * 1 mL in DMSO | ¥2832 | In-stock | |
1 mg | ¥1400 | In-stock | |
5 mg | ¥3500 | In-stock | |
10 mg | ¥5000 | In-stock | |
50 mg | ¥15000 | In-stock | |
100 mg | ¥21000 | In-stock | |
200 mg | 询价 | ||
500 mg | 询价 |
* Please select Quantity before adding items.
PSI-697 相关产品
•相关化合物库:
- Clinical Compound Library Plus
- Bioactive Compound Library Plus
生物活性 |
PSI-697 is an oral P-selectin inhibitor with an IC50 of 125 μM[1]. |
IC50 & Target |
IC50: 125 μM (P-selectin)[1] |
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体外研究 (In Vitro) |
PSI-697 inhibits the binding of a soluble human P-selectin to PSGL-1, in a reproducible concentration-dependent manner inhibiting 50% of binding at a concentration of 125 μM in vitro[1]. 上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only. |
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体内研究 (In Vivo) |
PSI-697 (0-50 mg/kg; p.o.) significantly reduces the number of rolling leukocytes by 39% versus vehicle control[1]. 上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only.
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Clinical Trial |
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分子量 |
367.83 |
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Formula |
C21H18ClNO3 |
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CAS 号 |
851546-61-7 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:
DMSO : ≥ 45.8 mg/mL (124.51 mM) * “≥” means soluble, but saturation unknown. 配制储备液
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请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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