SB-429201

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上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

SB-429201 

SB-429201 是一种有效的选择性 HDAC1 (IC50~1.5 μM)。SB-429201 对 HDAC1 抑制的偏好至少是 HDAC3 和 HDAC8 的 20 倍。

SB-429201

SB-429201 Chemical Structure

CAS No. : 1027971-34-1

规格 价格 是否有货 数量
5 mg ￥4200 In-stock
10 mg ￥6700 In-stock
25 mg ￥13500 In-stock
50 mg   询价  
100 mg   询价  

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SB-429201 相关产品

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生物活性

SB-429201 is a potent and selective HDAC1 (IC50~1.5 μM). SB-429201 displays at least a 20-fold preference for HDAC1 inhibition over HDAC3 and HDAC8[1][2].

IC50 & Target[1]

HDAC3

1.5 μM (IC50)

分子量

436.50

Formula

C28H24N2O3
CAS 号

1027971-34-1
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
参考文献

  • [1]. Hu E, et al. Identification of novel isoform-selective inhibitors within class I histone deacetylases. J Pharmacol Exp Ther. 2003;307(2):720-728.

    [2]. Bieliauskas AV, Pflum MK. Isoform-selective histone deacetylase inhibitors. Chem Soc Rev. 2008;37(7):1402-1413.

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