Monoamine oxidase/Aromatase-IN-1

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上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

Monoamine oxidase/Aromatase-IN-1 

Monoamine oxidase/Aromatase-IN-1 (compound 2q) 是一种高效的单胺氧化酶 (MAO) 和芳香化酶 (aromatase) 抑制剂，对 MAO-B 和芳香化酶的 IC50 分别为 39 nM 和 31 nM。Monoamine oxidase/Aromatase-IN-1 可用于神经系统疾病和乳腺癌的研究。

Monoamine oxidase/Aromatase-IN-1

Monoamine oxidase/Aromatase-IN-1 Chemical Structure

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生物活性

Monoamine oxidase/Aromatase-IN-1 (compound 2q) is a highly potent monoamine oxidase (MAO) and aromatase dual inhibitor with IC50s of 39 nM and 31 nM for MAO-B and aromatase, respectively. Monoamine oxidase/Aromatase-IN-1 can be used for researching neurological disorder and breast cancer[1].

IC50 & Target[1]

MAO-B

39 nM (IC50)

分子量

369.44

Formula

C19H19N3O3S
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Evren AE, et al. Synthesis of novel thiazolyl hydrazone derivatives as potent dual monoamine oxidase-aromatase inhibitors. Eur J Med Chem. 2022;229:114097.

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